Raw Local Anesthetic Agents Pharmaceutical Materials Procaine HCL CAS51-05-8

CAS : 51-05-8
MF: C13H21ClN2O2
MW: 272.77
EINECS: 200-077-2
Appearance:fine white crystalline powder, odorless, bitter, easily soluble in water, soluble in

ethanol, soluble in chloroform,

Procaine HCL is an anesthetic,non-toxic, free of side effects. Procaine HCL when injected into the muscles acts as an anesthetic but when taken orally in a complexed form procaine acts as a vitamin. Procaine HCl solutions, used as anesthetics, are tradenamed Novocaine.

Procaine HCl (procaine hydrochloride) is the active ingredient in Gerovital H3 (GH3) and in the Vitacels 3

through 8. Procaine HCl is broken down rapidly by enzymes in the blood stream into PABA and DEAE. The PABA and DEAE are rapidly conjugated and removed from the blood and excreted from the body.

Because of this procaine HCl and its breakdown products (metabolites) are unable to get into the cells in

any great quantity to produce benefits. Procaine HCl will produce some benefits by itself, but they are very limited.

Procaine HCl when combined with biologically active acids(1) such as folic acid, biotin,ascorbic acid,

pantothenic acid, citric acid and many other acids such as amino acids etc., acts as a vitamin or food

supplement. The vitamin acids and other biologically active acids when complexed with the procaine HCl

molecule protect the procaine from the enzymes in the blood allowing the procaine to enter the cells.

These vitamin complexes help the cells assimilate and utilize nutrients more efficiently. These complexed

procaine compounds named Vitacel (Vital Cell).

Procaine hcl, when taken orally, enters the body by being mainly absorbed through the villi in the small

intestine. Experiments show that the bulk of the procaine HCl enters the bloodstream molecularly intact. In the blood stream procaine HCl is rapidly hydrolyzed by the enzyme pseudo-cholinesterase into PABA and DEAE the two components of the procaine molecule. These metabolites are removed by the liver, chemically changed, and excreted in the urine.

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